E. F. Sagitova, D. N. Tomilin, O. V. Petrova, A. B. Budaev, L. N. Sobenina, B. A. Trofimov, G. Q. Yang, R. Hu, “Acetylene based short route from 2,2,6,6-tetramethylpiperidin-4-one oxime to 2-(pyrazol-5-yl)-4,5,6,7-tetrahydropyrrolo[3,2-c]pyridines”, Mendeleev Commun., 29:6 (2019), 658

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Mendeleev Communications, 2019, Volume 29, Issue 6, Pages 658–660
DOI: https://doi.org/10.1016/j.mencom.2019.11.018 (Mi mendc1621)

This article is cited in 3 scientific papers (total in 3 papers)

Communications

Acetylene based short route from 2,2,6,6-tetramethylpiperidin-4-one oxime to 2-(pyrazol-5-yl)-4,5,6,7-tetrahydropyrrolo[3,2-c]pyridines

E. F. Sagitova^a, D. N. Tomilin^a, O. V. Petrova^a, A. B. Budaev^a, L. N. Sobenina^a, B. A. Trofimov^a, G. Q. Yang^b, R. Hu^b

^a A.E. Favorsky Irkutsk Institute of Chemistry, Siberian Branch of the Russian Academy of Sciences, Irkutsk, Russian Federation
^b Institute of Chemistry, Chinese Academy of Sciences, Beijing, China

Full-text PDF (200 kB) Citations (3) Supplementary materials

DOI: https://doi.org/10.1016/j.mencom.2019.11.018

Graphic abstract: Acetylene based short route from 2,2,6,6-tetramethylpiperidin-4-one oxime to 2-(pyrazol-5-yl)-4,5,6,7-tetrahydropyrrolo[3,2-<i>c</i>]pyridines

Abstract: Pharmaceutically relevant substituted 2-(pyrazol-5-yl)-4,5,6,7-tetrahydropyrrolo [3,2-c]pyridines have been assembled in good to excellent yields via the reaction of 2,2,6,6-tetramethylpiperidin-4-one oxime with acetylene, cross-coupling of the resulting 4,4,6,6-tetramethyl-4,5,6,7 tetrahydropyrrolo[3,2-c]pyridines with aroylbromoacetylenes, and reaction of the formed 2-(aroylethynyl)-4,4,6,6-tetramethyl-4,5,6,7-tetrahydropyrrolo[3,2-c]pyridines with hydrazine.

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Document Type: Article

Language: English

*Supplementary materials:*
		Supplementary_data_1.pdf	(2.2 Mb)

Citation: E. F. Sagitova, D. N. Tomilin, O. V. Petrova, A. B. Budaev, L. N. Sobenina, B. A. Trofimov, G. Q. Yang, R. Hu, “Acetylene based short route from 2,2,6,6-tetramethylpiperidin-4-one oxime to 2-(pyrazol-5-yl)-4,5,6,7-tetrahydropyrrolo[3,2-c]pyridines”, Mendeleev Commun., 29:6 (2019), 658–660

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https://www.mathnet.ru/eng/mendc1621

https://www.mathnet.ru/eng/mendc/v29/i6/p658

This publication is cited in the following 3 articles:

Citing articles in Google Scholar: Russian citations, English citations
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