Ya. Yu. Shmoylova, Yu. A. Kovygin, E. A. Kosheleva, Kh. S. Shikhaliev, I. V. Ledenyova, M. A. Prezent, “Efficient synthesis of tetrahydro-1H-pyrazolo[3,4-b]pyridines based on the recyclization of N-arylitaconimides with aminopyrazoles”, Mendeleev Commun., 32:5 (2022), 688

Mendeleev Communications

RUS ENG

JOURNALS PEOPLE ORGANISATIONS CONFERENCES SEMINARS VIDEO LIBRARY PACKAGE AMSBIB

JavaScript is disabled in your browser. Please switch it on to enable full functionality of the website

	General information
	Latest issue
	Archive

	Search papers
	Search references

	RSS
	Latest issue
	Current issues
	Archive issues
	What is RSS

Mendeleev Commun.:
Year:
Volume:
Issue:
Page:
	Find

Personal entry:
Login:
Password:
	Save password
	Enter
	Forgotten password?
	Register

Mendeleev Communications, 2022, Volume 32, Issue 5, Pages 688–690
DOI: https://doi.org/10.1016/j.mencom.2022.09.041 (Mi mendc769)

This article is cited in 8 scientific papers (total in 8 papers)

Communications

Efficient synthesis of tetrahydro-1H-pyrazolo[3,4-b]pyridines based on the recyclization of N-arylitaconimides with aminopyrazoles

Ya. Yu. Shmoylova^a, Yu. A. Kovygin^a, E. A. Kosheleva^a, Kh. S. Shikhaliev^a, I. V. Ledenyova^a, M. A. Prezent^b

^a Department of Chemistry, Voronezh State University, Voronezh, Russian Federation
^b N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Moscow, Russian Federation

Full-text PDF (192 kB) Citations (8) Supplementary materials

DOI: https://doi.org/10.1016/j.mencom.2022.09.041

Graphic abstract: Efficient synthesis of tetrahydro-1<i>H</i>-pyrazolo[3,4-<i>b</i>]pyridines based on the recyclization of <i>N</i>-arylitaconimides with aminopyrazoles

Abstract: New polyfunctional hydrogenated pyrazolo[3,4-b]pyridines were obtained by the chemoselective reaction between N-arylitaconimides and 5-aminopyrazoles. The transformation is the cascade reaction including Michael addition at the active double bond of the itaconimide followed by the intramolecular transamidation and recyclization.

Keywords: pyrazolo[3,4-b]pyridines, itaconimides, 5-aminopyrazoles, recyclization, chemoselectivity, heterocyclization.

Bibliographic databases:

Document Type: Article

Language: English

*Supplementary materials:*
		Supplementary_data_1.pdf	(4.2 Mb)

Citation: Ya. Yu. Shmoylova, Yu. A. Kovygin, E. A. Kosheleva, Kh. S. Shikhaliev, I. V. Ledenyova, M. A. Prezent, “Efficient synthesis of tetrahydro-1H-pyrazolo[3,4-b]pyridines based on the recyclization of N-arylitaconimides with aminopyrazoles”, Mendeleev Commun., 32:5 (2022), 688–690

Linking options:

https://www.mathnet.ru/eng/mendc769

https://www.mathnet.ru/eng/mendc/v32/i5/p688

This publication is cited in the following 8 articles:

Citing articles in Google Scholar: Russian citations, English citations
Related articles in Google Scholar: Russian articles, English articles

Registration to the website

Logotypes